Department Researches & Publications

Faculty of Pharmacy

Assiut University

Department of Medicinal Chemistry

Researches

Our research spans a wide range from basic organic synthesis, drug design and development, structure elucidation of newly synthesized compound and natural products.

The research focuses on the following strategic Research Themes:

  • Design and synthesis of new chemical entities.
  • Computer aided drug design studies.
  • Structure-Activity relationship studies.
  • Combinatorial chemistry.
  • Prod rugs developments.
  • Analytical methods for bioavailability and metabolic studies.

Research within these Themes is carried out in multidisciplinary groupings focused on the discovery of novel techniques and/or enhancement of the already existing ones. At the department of Medicinal Pharmacy, We have major national and international collaborative research projects and a significant output of research publications in high-ranking journals. Our academic collaborators include many Universities in USA, Canada, Japan, and a number of major European universities.

 

 

# Title Research Year
81 Cu (I) Catalyzed Alkyne-Azide 1,3-Dipolar Cycloaddition (CuAAC): Synthesis of 17α-[1-(Substituted Phenyl)-1,2,3-Triazol-4-yl]-19-Nortestosterone-17β-yl Acetates Targeting Progestational and Antipro-Liferative Activities 2015
82 Lipases-catalyzed enantioselective kinetic resolution of alcohols 2015
83 Cu (I) Catalyzed Alkyne-Azide 1,3-Dipolar Cycloaddition (CuAAC): Synthesis of 17α-[1-(Substituted Phenyl)-1,2,3-Triazol-4-yl]-19-Nortestosterone-17β-yl Acetates Targeting Progestational and Antipro-Liferative Activities 2015
84 Lipases-catalyzed enantioselective kinetic resolution of alcohols 2015
85 Cu (I) Catalyzed Alkyne-Azide 1,3-Dipolar Cycloaddition (CuAAC): Synthesis of 17α-[1-(Substituted Phenyl)-1,2,3-Triazol-4-yl]-19-Nortestosterone-17β-yl Acetates Targeting Progestational and Antipro-Liferative Activities 2015
86 Optogenetic Inhibitor of the Transcription Factor CREB 2015
87 Lipases-catalyzed enantioselective kinetic resolution of alcohols 2015
88 Optimizing the Photocontrol of bZIP Coiled Coils with Azobenzene Crosslinkers: Role of the Crosslinking Site 2015
89 Cu (I) Catalyzed Alkyne-Azide 1,3-Dipolar Cycloaddition (CuAAC): Synthesis of 17α-[1-(Substituted Phenyl)-1,2,3-Triazol-4-yl]-19-Nortestosterone-17β-yl Acetates Targeting Progestational and Antipro-Liferative Activities 2015
90 Lipases-catalyzed enantioselective kinetic resolution of alcohols 2015